
PHARMACEUTICALS
AFFECTING THE
AUTONOMIC NERVOUS SYSTEM
AND
THE NEUROMUSCULAR JUNCTION
SYMPATHETIC NERVOUS SYSTEM
Direct - acting sympathomimetics
Non-selective:
norepinephrine (Levophed)
epinephrine chloride (Adrenalin)
Mixed Alpha:
norepinephrine (Levophed)
epinephrine chloride (Adrenalin)
Alpha1 agonists:
methoxamine HCl (Vasoxyl)
phenylephrine (Neo-Synephrine)
ephedrine
phenylpropanolamine (Propagest)
Alpha2 agonists:
clonidine (Catapres)
Mixed Beta agonists:
isoproterenol HCl (Isuprel)
epinephrine chloride (Adrenalin)
Beta1 agonist activity:
norepinephrine (Levophed)
dobutamine (Dobutrex)
dopamine HCl (Intropin; Dopastat)
Beta2 agonists:
albuterol sulfate (Proventil; Ventolin)
metaproterenol sulfate (Metaprel)
terbutaline sulfate (Bricanyl; Brethine)
ritodrine HCl (Yutopar)
Indirect - acting Sympathomimetics
tyramine
ephedrine
amphetamine (Benzedrine)
phenylpropanolamine (Propagest)
Catecholamine uptake inhibitors
cocaine
tricyclic antidepressants
Alpha-adrenergic antagonists
Non-selective:
phenoxybenzamine HCl (Dibenzyline)
phentolamine mesylate (Regitine)
ergot alkaloids, ergotamine
Alpha1 antagonists:
prazosin (Minipress)
terazocin (Hytrin)
Alpha2 antahonists:
yohimbine (Yocon, Yohimex)
Beta-adrenergic antagonists
Non-selective:
propranolol (Inderal)
pindolol (Visken)
nadolol (Corgard)
timolol maleate (Blocadrin)
Beta1 antagonists:
metoprolol tartrate (Lopressor)
acebutolol HCl (Sectral)
atenolol (Tenormin)
esmolol HCl (Brevibloc)
Mixed alpha/beta antagonsits:
labetalol HCl (Trandate; Normodyne)
Reducers of Central Sympathetic Outflow
methyldopa (Aldomet)
clonidine HCl (Catapres)
guanfacine HCl (Tenex)
guanabenz acetate (Wytensin)
Blockers of Norepinephrine Release
bretylium sulfate (Bretylol)
guanadrel sulfate (Hylorel)
guanethidine sulfate (Ismelin)
PARASYMPATHETIC NERVOUS SYSTEM
Parasympathomimetics
Muscarinic agonists:
acetylcholine chloride (Miochol)
carbachol Cl (Miostat; Carbacel)
methacholine (Provocholine)
bethanechol (Urecholine; Myotonachol)
pilocarpine HCl (Akarpine; Pilocar)
muscarine
Nicotinic agonists:
nicotine (Habitrol; Nicorette)
Cholinesterase inhibitors
physostigmine, eserine (Antilirium)
edrophonium Cl (Tensilon; Reversol)
neostigmine Br (Prostigmin)
pyridostigmine Br (Mestinon; Regonol)
tacrine HCl (Cognex)
DFP; isoflurophate (Floropryl)
echothiophate (Phospholine)
Cholinesterase Regenerator:
pralidoxime Cl; 2-PAM (Protopam)
Muscarinic blocking drugs
atropine sulfate (Isopto Atropine)
scopolamine HBr (Hyosol; Hyoscine)
ipratropium Br (Atrovent)
tropicamide (Mydriacyl)
trihexyphenidyl (Artane)
atropine methylnitrate (Metropine)
glycopyrrolate (Robinul)
propantheline Br (Pro-Banthine)
Nicotinic blocking drugs (ganglionic)
hexamethonium
trimethaphan camsylate (Arfonad)
mecamylamine HCl (Inversine)
NEUROMUSCULAR JUNCTION
Neuromuscular blocking drugs
hemicholinium
botulinum toxin
Non-depolarizing
d-tubocurarine (Tubarine)
pancuronium Br (Pavulon)
atracurium besylate (Tracrium)
vecuronium Br (Norcuron)
Depolarizing
succinylcholine (Anectine; Quelicin)
If you have comments or suggestions, email koritnik@ipfw.edu
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