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DRUGS BLOCKING AUTACOID RELEASE OR |
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DRUGS MIMICING AUTACOID RELEASE
Histamine agonist
betazole (Histalog)
Prostaglandins
PGE1, alprostadil (Prostin VR)
PGE2, dinoprostone (Prostin E2)
PGF2alpha, dinoprost (Prostin F2 Alpha)
prostacyclin, PGI2
thromboxane, TXA2
DRUGS PREVENTING AUTACOID RELEASE / BLOCKING RESPONSE
Mast cell stabilizer
cromolyn sodium (Aarane; Intal)
Antihistamines
H1 Receptor antagonists:
tripelennamine (Pyribenzamine)
diphenhydramine (Benadryl)
dimenhydrinate (Dramamine)
chlorpheniramine (Chlor-Trimeton)
meclizine (Bonine; Antivert)
terfenadine (Seldane)
astemizole (Hismanal)
loratadine (Claritin)
cetirizine (Zyrtec)
clemastine (Tavist)
H2 Receptor antagonists:
cimetidine (Tagamet)
ranitidine (Zantac)
famotidine (Pepcid)
nizatidine (Axid)
Analgesic antipyretics
aspirin
acetaminophen (Tylenol)
ibuprofen (Motrin; Rufen)
NON-STEROIDAL ANTI-INFLAMMATORY DRUGS (NSAIDS)
aspirin
indomethacin (lndocin)
tolmetin (Tolectin)
sulindac (Anthrocine; Clinoril)
ibuprofen (Motrin)
naproxen (Naprosyn)
diflunisal (Dolobid)
ketoprofen (Orudis)
diclofenac (Voltaren)
nabumetone (Relafen)
flurbiprofen (Ansaid; Froben; Ocufen)
piroxicam (Feldane)
STEROIDAL ANTI-INFLAMMATORY DRUGS
prednisone (Deltasone; Meticorten)
DRUG TREATMENT FOR SPECIFIC CONDITIONS
Anti-rheumatic drugs
aurothioglucose (Solganal)
auranofin (Ridaural)
penicillamine (Cuprimine; Depen)
hydroxychloroquine (Plaquenil)
methotrexate (Rheumatrex)
Anti-gout drugs
colchicine
indomethacin (lndocin)
probenecid (Benemid)
sulfinpyrazone (Anturane)
allopurinol (Zyloprim)
Anti-asthmatic drugs
theophylline; aminophylline
epinephrine (Adrenalin) .
isoproterenol (Isuprel; Medihaler-Iso)
terbutaline (Bricanyl; Brethine)
albuterol; salbutamol (Proventil; Ventolin)
ipratropium (Atrovent) .
beclomethasone (Vanceril; Beclovent)
cromolyn sodium (Aarane; Intal)
nedocromil (Tilade)
zafirlukast (Accolate)
zileuton (Leutron)
DRUGS ALTERING THE IMMUNE RESPONSE
immunoglobulins (several)
prednisone (Deltasone; Orasone)
azathioprim (Imuran)
cyclophosphamide (Cytoxan; Neospar)
cyclosporine (Sandimmune)
methotrexate (Folex; Mexate)
cytarabine; ara-C (Citosar-U)
vincristine (Oncovin)
If you have comments or suggestions, email koritnik@ipfw.edu